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受容体 (リガンド) | GlyRTooltip Glycine receptor/ja |
- 陽性モジュレーター: アルコール (例えば、 brometone/ja, クロロブタノール(クロレトン), エタノール(アルコール), tert-ブタノール (2M2P), tribromoethanol/ja, trichloroethanol/ja, trifluoroethanol/ja)
- Alkylbenzene sulfonate/ja
- Anandamide/ja
- Barbiturate/ja (例えば、pentobarbital/ja, sodium thiopental/ja)
- Chlormethiazole/ja
- D12-116/ja
- Dihydropyridine/ja (例えば、 nicardipine/ja)
- Etomidate/ja
- Ginseng/ja 成分 (例えば、ginsenoside/ja (例えば、ginsenoside-Rf/ja))
- グルタミン酸 (glutamate)
- Ivermectin/ja
- Ketamine/ja
- Neuroactive steroid/ja (例えば、alfaxolone/ja, プレグネノロン(エルタノロン), pregnenolone acetate/ja, minaxolone/ja, ORG-20599/ja)
- Nitrous oxide/ja
- Penicillin G/ja
- Propofol/ja
- Tamoxifen/ja
- Tetrahydrocannabinol/ja
- Triclofos/ja
- Tropeine/ja (例えば、atropine/ja, bemesetron/ja, cocaine/ja, LY-278584/ja, tropisetron/ja, zatosetron/ja)
- 揮発性物質/gas/ja (例えば、chloral hydrate/ja, chloroform/ja, desflurane/ja, ジエチルエーテル(エーテル), enflurane/ja, halothane/ja, isoflurane/ja, methoxyflurane/ja, sevoflurane/ja, toluene/ja, トリクロロエタン(メチルクロロホルム), trichloroethylene/ja)
- Xenon/ja
- 亜鉛
- 陰性モジュレーター: Amiloride/ja
- Benzodiazepine/ja (例えば、bromazepam/ja, clonazepam/ja, diazepam/ja, flunitrazepam/ja, flurazepam/ja)
- Corymine/ja
- Cyanotriphenylborate/ja
- Daidzein/ja
- Dihydropyridine/ja (例えば、nicardipine/ja, nifedipine/ja, nitrendipine/ja)
- Furosemide/ja
- Genistein/ja
- イチョウ 成分 (例えば、bilobalide/ja, ginkgolide/ja (例えば、ginkgolide A/ja, ginkgolide B/ja, ginkgolide C/ja, ginkgolide J/ja, ginkgolide M/ja))
- Imipramine/ja
- NBQX/ja
- Neuroactive steroid/ja (例えば、3α-androsterone sulfate/ja, 3β-androsterone sulfate/ja, デオキシコルチコステロン, DHEA sulfate/ja, pregnenolone sulfate/ja, progesterone/ja)
- Opioid/ja (例えば、codeine/ja, dextromethorphan/ja, dextrorphan/ja, levomethadone/ja, levorphanol/ja, morphine/ja, oripavine/ja, pethidine/ja, thebaine/ja)
- Picrotoxin/ja (すなわち、picrotin/ja と picrotoxinin/ja)
- PMBA
- Riluzole/ja
- Tropeine/ja (例えば、bemesetron/ja, LY-278584/ja, tropisetron/ja, zatosetron/ja)
- Verapamil/ja
- 亜鉛
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NMDARTooltip N-Methyl-D-aspartate receptor/ja | |
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輸送体 (ブロッカーs) | GlyT1Tooltip Glycine transporter 1/ja | |
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GlyT2Tooltip Glycine transporter 2/ja | |
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カルシウム | VDCCsTooltip Voltage-dependent calcium channels/ja | |
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カリウム | VGKCsTooltip Voltage-gated potassium channels/ja | |
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IRKsTooltip Inwardly rectifying potassium channel/ja | |
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KCaTooltip Calcium-activated potassium channel/ja | |
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K2PsTooltip Tandem pore domain potassium channel/ja | |
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ナトリウム | VGSCsTooltip Voltage-gated sodium channels/ja | |
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ENaCTooltip Epithelial sodium channel/ja | |
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ASICsTooltip Acid-sensing ion channel/ja | |
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塩素 | CaCCsTooltip Calcium-activated chloride channel/ja | |
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CFTRTooltip Cystic fibrosis transmembrane conductance regulator/ja | |
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未整理 | |
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その他 | TRPsTooltip Transient receptor potential channels/ja | |
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LGICsTooltip Ligand gated ion channels/ja | |
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MRTooltip Mineralocorticoid receptor/ja | |
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CARTooltip Constitutive androstane receptor/ja | |
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PXRTooltip Pregnane X receptor/ja | |
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