Discovery and development of gliflozins/ja: Difference between revisions

Discovery and development of gliflozins/ja
Created page with "File:Mynd fyrir toflu1.png"
Created page with "{| class="wikitable" |- ! R !! IC<sub>50</sub> (nM) !! 活性 |- |align="center"| File:Bygging 1.png ||align="center"| 0.720 ||align="center"| ''試験管内''活性が向上* |- |align="center"| File:Bygging 2.png ||align="center"| 1.14 ||align="center"| ''試験管内''活性が向上* |- |align="center"| File:Bygging 3.png ||align="center"| 13.3 ||align="center"| 炭素数が増えるにつれて、IC-50値は変動 |- |align="center"| File:1-Methoxy-n-b..."
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[[File:Mynd fyrir toflu1.png]]
[[File:Mynd fyrir toflu1.png]]


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{| class="wikitable"
{| class="wikitable"
|-
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! R !! IC<sub>50</sub> (nM) !! Activity
! R !! IC<sub>50</sub> (nM) !! 活性
|-
|-
|align="center"| [[File:Bygging 1.png]] ||align="center"| 0.720 ||align="center"| ''in vitro'' activity improved*
|align="center"| [[File:Bygging 1.png]] ||align="center"| 0.720 ||align="center"| ''試験管内''活性が向上*
|-
|-
|align="center"| [[File:Bygging 2.png]] ||align="center"| 1.14 ||align="center"| ''in vitro'' activity improved*
|align="center"| [[File:Bygging 2.png]] ||align="center"| 1.14 ||align="center"| ''試験管内''活性が向上*
|-
|-
|align="center"| [[File:Bygging 3.png]] ||align="center"| 13.3 ||align="center"| As the number of carbons increases, the IC-50 value fluctuates
|align="center"| [[File:Bygging 3.png]] ||align="center"| 13.3 ||align="center"| 炭素数が増えるにつれて、IC-50値は変動
|-
|-
|align="center"| [[File:1-Methoxy-n-butane.png]] ||align="center"| 19.6 ||align="center"| ''in vitro'' activity decreased*
|align="center"| [[File:1-Methoxy-n-butane.png]] ||align="center"| 19.6 ||align="center"| ''試験管内''での''活性が低下*
|-
|-
|align="center"| [[File:Bygging 5.png]] ||align="center"| 21.2 ||align="center"| ''in vitro'' activity decreased*
|align="center"| [[File:Bygging 5.png]] ||align="center"| 21.2 ||align="center"| ''試験管内''での''活性が低下*
|}
|}
''*comparator to ethyl group (IC<sub>50</sub> = 16,7)''
''*エチル基との比較対象 (IC<sub>50</sub> = 16,7)''
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