Discovery and development of gliflozins/ja: Difference between revisions
Discovery and development of gliflozins/ja
Created page with "File:Mynd fyrir toflu1.png" |
Created page with "{| class="wikitable" |- ! R !! IC<sub>50</sub> (nM) !! 活性 |- |align="center"| File:Bygging 1.png ||align="center"| 0.720 ||align="center"| ''試験管内''活性が向上* |- |align="center"| File:Bygging 2.png ||align="center"| 1.14 ||align="center"| ''試験管内''活性が向上* |- |align="center"| File:Bygging 3.png ||align="center"| 13.3 ||align="center"| 炭素数が増えるにつれて、IC-50値は変動 |- |align="center"| File:1-Methoxy-n-b..." Tags: Mobile edit Mobile web edit |
||
Line 72: | Line 72: | ||
[[File:Mynd fyrir toflu1.png]] | [[File:Mynd fyrir toflu1.png]] | ||
{| class="wikitable" | {| class="wikitable" | ||
|- | |- | ||
! R !! IC<sub>50</sub> (nM) !! | ! R !! IC<sub>50</sub> (nM) !! 活性 | ||
|- | |- | ||
|align="center"| [[File:Bygging 1.png]] ||align="center"| 0.720 ||align="center"| '' | |align="center"| [[File:Bygging 1.png]] ||align="center"| 0.720 ||align="center"| ''試験管内''活性が向上* | ||
|- | |- | ||
|align="center"| [[File:Bygging 2.png]] ||align="center"| 1.14 ||align="center"| '' | |align="center"| [[File:Bygging 2.png]] ||align="center"| 1.14 ||align="center"| ''試験管内''活性が向上* | ||
|- | |- | ||
|align="center"| [[File:Bygging 3.png]] ||align="center"| 13.3 ||align="center"| | |align="center"| [[File:Bygging 3.png]] ||align="center"| 13.3 ||align="center"| 炭素数が増えるにつれて、IC-50値は変動 | ||
|- | |- | ||
|align="center"| [[File:1-Methoxy-n-butane.png]] ||align="center"| 19.6 ||align="center"| '' | |align="center"| [[File:1-Methoxy-n-butane.png]] ||align="center"| 19.6 ||align="center"| ''試験管内''での''活性が低下* | ||
|- | |- | ||
|align="center"| [[File:Bygging 5.png]] ||align="center"| 21.2 ||align="center"| '' | |align="center"| [[File:Bygging 5.png]] ||align="center"| 21.2 ||align="center"| ''試験管内''での''活性が低下* | ||
|} | |} | ||
''* | ''*エチル基との比較対象 (IC<sub>50</sub> = 16,7)'' | ||
<div lang="en" dir="ltr" class="mw-content-ltr"> | <div lang="en" dir="ltr" class="mw-content-ltr"> |