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Febuxostat/22/ja
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Revision as of 20:25, 22 April 2024 by
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(Created page with "{{Antigout preparations/ja}} {{Purinergics/ja}} {{Portal bar | Medicine}}")
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v
t
e
痛風
に使用される薬 (
M04
)
尿酸排泄促進薬
第一選択
Probenecid/ja
Sulfinpyrazone/ja
Benzbromarone/ja
Isobromindione/ja
第二選択
Amlodipine/ja
Atorvastatin/ja
Fenofibrate/ja
Guaifenesin/ja
Lesinurad/ja
‡
ロサルタン
キサンチンオキシダーゼ阻害剤
purine analogue/ja
Allopurinol/ja
#
Oxypurinol/ja
Tisopurine/ja
その他
フェブキソスタット
Inositol/ja
(
Phytic acid/ja
ミオイノシトール
)
Topiroxostat/ja
Mitotic inhibitor/ja
Colchicine/ja
その他
Cinchophen/ja
NSAIDs
(
aspirin/ja
を除く)
Sevelamer/ja
Urate oxidase/ja
(
Rasburicase/ja
Pegloticase/ja
)
#
WHO-EM
‡
Withdrawn
from market
Clinical trials
:
†
Phase III
§
Never to phase III
v
t
e
Purine receptor/ja
モジュレーター
受容体
(
リガンド
)
P0
(
adenine/ja
)
作用薬:
8-Aminoadenine/ja
Adenine/ja
P1
(
adenosine/ja
)
作用薬:
2-(1-ヘキシニル)-
N
-メチルアデノシン
2-Cl-IB-MECA/ja
2'-MeCCPA/ja
4'-O-β-D-グルコシル-9-O-(6''-デオキシサッカロシル)オリビル
5'-
N
-エチルカルボキサミドアデノシン
Adenosine/ja
ADP
AMP
Apadenoson/ja
ATL-146e/ja
ATP
BAY 60–6583/ja
Binodenoson/ja
Capadenoson/ja
CCPA
CGS-21680/ja
CP-532,903/ja
Evodenoson/ja
GR 79236/ja
LUF-5835/ja
LUF-5845/ja
N
6
-シクロペンチルアデノシン
Namodenoson/ja
Neladenoson dalanate/ja
Piclidenoson/ja
Regadenoson/ja
SDZ WAG 994/ja
Selodenoson/ja
Sonedenoson/ja
Tecadenoson/ja
UK-432,097/ja
拮抗薬:
7-Methylxanthine/ja
8-Chlorotheophylline/ja
8-Phenyl-1,3-dipropylxanthine/ja
8-Phenyltheophylline/ja
Acefylline/ja
Aminophylline/ja
ATL-444/ja
Bamifylline/ja
Cafedrine/ja
Caffeine/ja
Caffeine citrate/ja
Cartazolate/ja
CGH-2466/ja
CGS-15943/ja
Choline theophyllinate/ja
Ciforadenant/ja
CPX
CVT-6883/ja
Dimethazan/ja
DMPX/ja
DPCPX
Dyphylline/ja
Enprofylline/ja
Etazolate/ja
Fenethylline/ja
IBMX/ja
Isovaleric acid/ja
Istradefylline/ja
KF-26777/ja
MRE3008F20/ja
MRS-1220/ja
MRS-1334/ja
MRS-1706/ja
MRS-1754/ja
MRS-3777/ja
Paraxanthine/ja
Pentoxifylline/ja
Preladenant/ja
Propentofylline/ja
Proxyphylline/ja
PSB-10/ja
PSB-11/ja
PSB-36/ja
PSB-603/ja
PSB-788/ja
PSB-1115/ja
Reversine/ja
Rolofylline/ja
SCH-442,416/ja
SCH-58261/ja
Theacrine/ja
Theobromine/ja
Theodrenaline/ja
Theophylline/ja
Tozadenant/ja
Tracazolate/ja
VUF-5574/ja
ZM-241,385/ja
P2
(
nucleotide/ja
)
P2X
(
ATP
Tooltip Adenosine triphosphate/ja
)
作用薬:
2-Me-SATP
α,β-Me-ATP
Adenosine/ja
ADP
AMP
Ap4A
Ap5A
ATP
ATPγS
BzATP/ja
Cibacron blue/ja
CTP
D-β,γ-Me-ATP/ja
GTP
HT-AMP/ja
Ivermectin/ja
L-β,γ-Me-ATP/ja
MRS-2219/ja
PAPET-ATP/ja
UTP
亜鉛
拮抗薬:
5-BDBD/ja
A-317491/ja
A-438079/ja
A-740003/ja
A-804598/ja
A-839977/ja
AF-353/ja
AZ-10606120/ja
AZ-11645373/ja
BBG
Calcium/ja
Calmidazolium/ja
Chelerythrine/ja
Copper/ja
Emodin/ja
(
Rheum officinale
)
エヴァンス・ブルー
Gefapixant/ja
GW-791343/ja
HMA
Ip5I
isoPPADS/ja
JNJ-47965567/ja
KN-04/ja
KN-62/ja
Magnesium/ja
MRS-2159/ja
NF-023/ja
NF-110/ja
NF-157/ja
NF-279/ja
NF-449/ja
オピランセリン (VVZ-149)
Oxidized-ATP/ja
Phenol Red/ja
Phenolphthalein/ja
PPADS/ja
PPNDS/ja
PSB-12062/ja
Puerarin/ja
(
Radix puerariae/ja
)
Purotoxin 1/ja
RB-2
Ro 0437626/ja
Ro 51/ja
RO-3/ja
Sodium ferulate/ja
(
Angelica sinensis/ja
,
Ligusticum wallichii/ja
)
Suramin/ja
TC-P 262/ja
テトラメチルピラジン(リグストラジン)
(
Ligusticum wallichii/ja
)
TNP-ATP/ja
亜鉛
P2Y
Agonists:
2-Me-SADP
2-Me-SATP
2-Thio-UTP/ja
5-Br-UDP
5-OMe-UDP/ja
α,β-Me-ATP
Adenosine/ja
ADP
ADPβS
Ap3A
AR-C 67085MX/ja
ATP
ATPγS
CTP
dATP
Denufosol/ja
Diquafosol/ja
IDP
ITP
INS-365/ja
INS-37217/ja
MRS-2365/ja
MRS-2690/ja
MRS-2693/ja
MRS-2768/ja
MRS-2957/ja
MRS-4062/ja
NF-546/ja
PAPET-ATP/ja
PSB-0474/ja
PSB-1114/ja
UDP
UDPβS
UDP-ガラクトース
UDP-グルコース
UDP-N-アセチルグルコサミン
Up3U
UTP
UTPγS
拮抗薬:
2-Me-SAMP
A3P5PS/ja
AMPαS/ja
Ap4A
AR-C 66096/ja
AR-C 67085MX/ja
AR-C 69931MX/ja
AR-C 118925XX/ja
ATP
BzATP/ja
C1330-7/ja
Cangrelor/ja
Clopidogrel/ja
Elinogrel/ja
Ip5I
MRS-2179/ja
MRS-2211/ja
MRS-2279/ja
MRS-2395/ja
MRS-2500/ja
MRS-2578/ja
NF-157/ja
NF-340/ja
PIT
PPADS/ja
Prasugrel/ja
PSB-0739/ja
RB-2
Regrelor/ja
Suramin/ja
Ticagrelor/ja
Ticlopidine/ja
UDP
トランスポーター
(
ブロッカー
)
CNTs
Tooltip Concentrative nucleoside transporters/ja
6-Hydroxy-7-methoxyflavone/ja
Adenosine/ja
dMeThPmR/ja
Estradiol/ja
KGO-2142/ja
KGO-2173/ja
MeThPmR/ja
Phloridzin/ja
Progesterone/ja
ENTs
Tooltip Equilibrative nucleoside transporters/ja
Barbiturate/ja
Benzodiazepine/ja
Cilostazol/ja
Dilazep/ja
Dipyridamole/ja
Estradiol/ja
Ethanol/ja
Hexobendine/ja
NBMPR
Pentoxifylline/ja
Progesterone/ja
Propentofylline/ja
PMAT
Tooltip Plasma membrane monoamine transporter/ja
Decynium-22/ja
酵素
(
阻害剤
)
XO
Tooltip Xanthine oxidase/ja
Allopurinol/ja
Amflutizole/ja
Benzbromarone/ja
Caffeic acid/ja
Cinnamaldehyde/ja
Cinnamomum osmophloeum/ja
フェブキソスタット
Myo-inositol/ja
Kaempferol/ja
Myricetin/ja
Niraxostat/ja
Oxipurinol/ja
Phytic acid/ja
Pistacia integerrima/ja
Propolis/ja
Quercetin/ja
Tisopurine/ja
Topiroxostat/ja
その他
Aminopterin/ja
Azathioprine/ja
Methotrexate/ja
Mycophenolic acid/ja
Pemetrexed/ja
Pralatrexate/ja
その他多数
その他
前駆物質:
Adenine/ja
Adenosine/ja
AMP
ADP
ATP
Cytosine/ja
Cytidine/ja
CMP
CDP
CTP
Guanine/ja
Guanosine/ja
GMP
GDP
GTP
Hypoxanthine/ja
Inosine/ja
IMP
IDP
ITP
Ribose/ja
Uracil/ja
Uridine/ja
UMP
UDP
UTP
その他:
Chrysophanol/ja
(
rhubarb
)
こちらも参照:
受容体/シグナル伝達モジュレーター
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:
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