Translations:Dipeptidyl peptidase-4 inhibitor/6/en
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Examples
Drugs belonging to this class are:
- Sitagliptin (FDA approved 2006, marketed by Merck & Co. as Januvia)
- Vildagliptin (EU approved 2007, marketed in the EU by Novartis as Galvus)
- Saxagliptin (FDA approved in 2009, marketed as Onglyza)
- Linagliptin (FDA approved in 2011, marketed as Tradjenta by Eli Lilly and Company and Boehringer Ingelheim)
- Gemigliptin (approved in Korea in 2012, marketed by LG Life Sciences) Marketed as Zemiglo
- Anagliptin (approved in Japan as Suiny in 2012, marketed by Sanwa Kagaku Kenkyusho Co., Ltd. and Kowa Company, Ltd.)
- Teneligliptin (approved in Japan as Tenelia in 2012)
- Alogliptin (FDA approved 2013 as Nesina/ Vipidia, marketed by Takeda Pharmaceutical Company)
- Trelagliptin (approved for use in Japan as Zafatek/ Wedica in 2015)
- Omarigliptin (MK-3102) (approved as Marizev in Japan in 2015, developed by Merck & Co.; research showed that omarigliptin can be used as once-weekly treatment and generally well tolerated throughout the base and extension studies)
- Evogliptin (approved as Suganon/ Evodine for use in South Korea)
- Gosogliptin (approved as Saterex for use in Russia)
- Dutogliptin (PHX- 1149 free base, being developed by Phenomix Corporation), Phase III
- Retagliptin (SP-2086), approved in China.
- Denagliptin
- Cofrogliptin (HSK- 7653, compound 2)
- Fotagliptin
- Prusogliptin