Sitagliptin/ja: Difference between revisions
Sitagliptin/ja
Created page with "<!-- Legal status --> | legal_AU = S4 | legal_AU_comment = | legal_BR = <!-- OTC, A1, A2, A3, B1, B2, C1, C2, C3, C4, C5, D1, D2, E, F --> | legal_BR_comment = | legal_CA = <!-- OTC, Rx-only, Schedule I, II, III, IV, V, VI, VII, VIII --> | legal_CA_comment = | legal_DE = <!-- Anlage I, II, III or Unscheduled --> | legal_DE_comment = | legal_NZ = <!-- Class A, B, C --> | legal_NZ_comment = | legal_UK = POM | legal_UK_comment = | legal_US = Rx-only | legal_US_comment..." Tags: Mobile edit Mobile web edit |
Created page with "シタグリプチン" Tags: Mobile edit Mobile web edit |
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| legal_status = <!-- For countries not listed above --> | | legal_status = <!-- For countries not listed above --> | ||
<!-- Pharmacokinetic data --> | <!-- Pharmacokinetic data --> | ||
| bioavailability = 87% | | bioavailability = 87% | ||
| protein_bound = 38% | | protein_bound = 38% | ||
| metabolism = [[Liver]] ([[CYP3A4]]- | | metabolism = [[Liver/ja|肝臓]] ([[CYP3A4/ja|CYP3A4]]- と [[CYP2C8/ja|CYP2C8]]-介在) | ||
| metabolites = | | metabolites = | ||
| onset = | | onset = | ||
| elimination_half-life = 8 to 14 h | | elimination_half-life = 8 to 14 h | ||
| duration_of_action = | | duration_of_action = | ||
| excretion = [[Kidney]] (80%) | | excretion = [[Kidney/ja]] (80%) | ||
<!-- Identifiers --> | <!-- Identifiers --> | ||
| index2_label = as salt | | index2_label = as salt | ||
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| NIAID_ChemDB = | | NIAID_ChemDB = | ||
| PDB_ligand = | | PDB_ligand = | ||
| synonyms = | | synonyms = | ||
<!-- Chemical and physical data --> | <!-- Chemical and physical data --> | ||
| IUPAC_name = (''R'')-4-oxo-4-[3-(trifluoromethyl)-5,6-dihydro[1,2,4]triazolo[4,3-''a'']pyrazin-7(8''H'')-yl]-1-(2,4,5-trifluorophenyl)butan-2-amine | | IUPAC_name = (''R'')-4-oxo-4-[3-(trifluoromethyl)-5,6-dihydro[1,2,4]triazolo[4,3-''a'']pyrazin-7(8''H'')-yl]-1-(2,4,5-trifluorophenyl)butan-2-amine | ||
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| specific_rotation = | | specific_rotation = | ||
}} | }} | ||
<div lang="en" dir="ltr" class="mw-content-ltr"> | <div lang="en" dir="ltr" class="mw-content-ltr"> | ||