Translations:Angiotensin II receptor blocker/25/en
The ratios of AT1 to AT2 in binding affinities of the specific ARBs are shown as follows. However, AT1 affinity vs AT2 is not a meaningful indicator of blood pressure response.
- Losartan – 1000-fold
- Telmisartan – 3000-fold
- Irbesartan – 8500-fold
- Candesartan – greater than 10000-fold
- Olmesartan – 12500-fold
- Valsartan – 30000-fold
- Saprisartan – ???