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Discovery and development of gliflozins/29/ja
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Revision as of 15:48, 14 February 2024 by
Fire
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(Created page with "{| class="wikitable" |- ! R !! IC<sub>50</sub> (nM) !! 活性 |- |align="center"|
File:Bygging 1.png
||align="center"| 0.720 ||align="center"| ''試験管内''活性が向上* |- |align="center"|
File:Bygging 2.png
||align="center"| 1.14 ||align="center"| ''試験管内''活性が向上* |- |align="center"|
File:Bygging 3.png
||align="center"| 13.3 ||align="center"| 炭素数が増えるにつれて、IC-50値は変動 |- |align="center"| File:1-Methoxy-n-b...")
(diff) ← Older revision | Latest revision (diff) | Newer revision → (diff)
R
IC
50
(nM)
活性
0.720
試験管内
活性が向上*
1.14
試験管内
活性が向上*
13.3
炭素数が増えるにつれて、IC-50値は変動
19.6
試験管内
での
活性が低下*
21.2
試験管内
での
活性が低下*
*エチル基との比較対象 (IC
50
= 16,7)