Translations
:
GLP-1 receptor agonist/24/en
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v
t
e
Oral
diabetes medication
,
insulins
and
insulin analogs
, and other drugs used in diabetes (
A10
)
Insulins
/
insulin analogs
fast-acting
Insulin aspart
Insulin glulisine
Insulin lispro
short-acting
Regular insulin
#
long-acting
Insulin detemir
#
Insulin glargine
#
(
+lixisenatide
)
NPH insulin
Lente insulin
‡
Ultralente insulin
‡
ultra-long-acting
Insulin degludec
#
(
+insulin aspart
,
+liraglutide
)
Insulin icodec
†
(
+semaglutide
)
inhalable
Exubera
‡
Afrezza
#
WHO-EM
‡
Withdrawn
from market
Clinical trials
:
†
Phase III
§
Never to phase III
Non-insulins
Insulin sensitizers
Biguanides
Buformin
‡
Metformin
#
Phenformin
‡
TZDs
/"glitazones" (
PPAR
)
Ciglitazone
§
Darglitazone
§
Englitazone
§
Lobeglitazone
Netoglitazone
§
Pioglitazone
Rivoglitazone
†
Rosiglitazone
Troglitazone
‡
Dual PPAR agonists
Aleglitazar
†
Muraglitazar
§
Saroglitazar
Tesaglitazar
§
Amylin
analogs and
DACRAs
Cagrilintide
§
Pramlintide
Secretagogues
K
+
ATP
Sulfonylureas
1st generation
:
Acetohexamide
Carbutamide
Chlorpropamide
Glycyclamide
Metahexamide
Tolazamide
Tolbutamide
2nd generation
:
Glibenclamide (glyburide)
Glibornuride
Glicaramide
Gliclazide
#
Glimepiride
Glipizide
Gliquidone
Glisoxepide
Glyclopyramide
Meglitinides
/"glinides"
Mitiglinide
Nateglinide
Repaglinide
GLP-1 receptor agonists
Albiglutide
‡
Danuglipron
†
Dulaglutide
Exenatide
Liraglutide
Lixisenatide
Orforglipron
§
Semaglutide
Taspoglutide
†
GLP1 poly-agonist peptides
Mazdutide
(GLP-1/
GCGR
)
Retatrutide
§
(GLP-1/GIP/GCGR)
Tirzepatide
(GLP-1/GIP)
DPP-4 inhibitors
/"gliptins"
Alogliptin
Anagliptin
Evogliptin
Garvagliptin
Gemigliptin
Gosogliptin
Linagliptin
Melogliptin
Omarigliptin
Saxagliptin
Sitagliptin
Teneligliptin
Trelagliptin
Vildagliptin
Other
Aldose reductase inhibitors
Epalrestat
Fidarestat
§
Ranirestat
†
Tolrestat
‡
Zenarestat
§
Alpha-glucosidase inhibitors
Acarbose
Miglitol
Voglibose
SGLT2 inhibitors
/"gliflozins"
Canagliflozin
Dapagliflozin
Empagliflozin
#
Ertugliflozin
Ipragliflozin
Luseogliflozin
Remogliflozin
§
Sergliflozin
§
Sotagliflozin
Tofogliflozin
†
Velagliflozin
Other
Benfluorex
‡
Bromocriptine
Imeglimin
Combinations
Alogliptin/metformin
Canagliflozin/metformin
Cagrilintide/semaglutide
§
Dapagliflozin/metformin
Dapagliflozin/saxagliptin
Dapagliflozin/saxagliptin/metformin
Empagliflozin/linagliptin
Empagliflozin/metformin
Gemigliptin/rosuvastatin
Glibenclamide (glyburide)/metformin
Glimepiride/rosiglitazone
Linagliptin/metformin
Metformin/acarbose
Metformin/ertugliflozin
Metformin/evogliptin
Metformin/gemigliptin
Metformin/repaglinide
Metformin/sulfonylureas
Metformin/teneligliptin
Phenformin/sulfonylureas
Pioglitazone/alogliptin
Pioglitazone/glimepiride
Pioglitazone/metformin
Pioglitazone/sitagliptin
Rosiglitazone/metformin
Saxagliptin/metformin
Sitagliptin/dapagliflozin
Sitagliptin/ertugliflozin
Sitagliptin/metformin
Sitagliptin/simvastatin
Vildagliptin/metformin
#
WHO-EM
‡
Withdrawn
from market
Clinical trials
:
†
Phase III
§
Never to phase III
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