Translations
:
Ethyl eicosapentaenoic acid/28/en
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v
t
e
Lipid-lowering agents
(
C10
)
GI tract
Cholesterol absorption inhibitors
,
NPC1L1
Ezetimibe
SCH-48461
Bile acid sequestrants
/
resins
(
LDL
)
Colesevelam
Colestilan
Colestipol
Colestyramine
Colextran
Soluble fiber
such as
psyllium
and
glucomannan
Liver
Statins
(
HMG-CoA reductase
,
LDL
)
Atorvastatin
Cerivastatin
‡
Fluvastatin
Lovastatin
Mevastatin
Pitavastatin
Pravastatin
Rosuvastatin
Simvastatin
#
Niacin and derivatives (
HDL
and
LDL
)
Acipimox
Aluminium nicotinate
Niacin
Niceritrol
Nicofuranose
Nicotinyl alcohol
MTTP
inhibitors (
VLDL
)
Dirlotapide
Lomitapide
Mitratapide
ATP citrate lyase
inhibitors (
LDL
)
Bempedoic acid
Thyromimetics
(VLDL)
Dextrothyroxine
‡
Resmetirom
Blood vessels
PPAR agonists
(LDL)
Fibrates
Aluminium clofibrate
Bezafibrate
Choline fenofibrate
Ciprofibrate
Clinofibrate
Clofibrate
‡
Clofibride
Etofibrate
Fenofibrate
Gemfibrozil
Nafenopin
Pemafibrate
Ronifibrate
Simfibrate
Others
GW501516
§
CETP inhibitors
(
HDL
)
Anacetrapib
†
Dalcetrapib
§
Evacetrapib
§
Obicetrapib
†
Torcetrapib
§
PCSK9 inhibitors
(
LDL
)
Alirocumab
Bococizumab
Evolocumab
Inclisiran
ANGPTL3
inhibitors (
LDL
/
HDL
)
Evinacumab
Combinations
Amlodipine/atorvastatin
Bempedoic acid/ezetimibe
Ezetimibe/atorvastatin
Ezetimibe/rosuvastatin
Ezetimibe/simvastatin
Fenofibrate/pravastatin
Fenofibrate/simvastatin
Niacin/laropiprant
Niacin/lovastatin
Niacin/simvastatin
Other
Alipogene tiparvovec
Azacosterol
Azalanstat
Benfluorex
‡
Darapladib
§
Lapaquistat
§
Magnesium pyridoxal 5-phosphate glutamate
Meglutol
Mipomersen
Omega-3-triglycerides
Policosanol
Probucol
Tiadenol
Triparanol
‡
Volanesorsen
#
WHO-EM
‡
Withdrawn
from market
Clinical trials
:
†
Phase III
§
Never to phase III
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