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:
Insulin analog/22/ja
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v
t
e
経口
糖尿病治療薬
、
インスリン
製剤および
インスリンアナログ
製剤、糖尿病に用いられるその他の薬剤(
A10
)
インスリン
/
インスリンアナログ
超速効型
Insulin aspart/ja
Insulin glulisine/ja
Insulin lispro/ja
速効型
Regular insulin/ja
#
長時間作用型
Insulin detemir/ja
#
インスリングラルギン
#
(
+リキセナチド
)
NPH insulin/ja
Lente insulin/ja
‡
Ultralente insulin/ja
‡
超長時間作業型
Insulin degludec/ja
#
(
+インスリンアスパルト
,
+リラグルチド
)
Insulin icodec/ja
†
(
+セマグルチド
)
吸入可能
Exubera
‡
Afrezza
#
WHO-EM
‡
Withdrawn
from market
Clinical trials
:
†
Phase III
§
Never to phase III
非インスリン
インスリン感作薬
ビグアナイド
Buformin/ja
‡
メトホルミン
#
Phenformin/ja
‡
TZD
/"グリタゾン" (
PPAR
)
Ciglitazone/ja
§
Darglitazone/ja
§
Englitazone/ja
§
Lobeglitazone/ja
Netoglitazone/ja
§
Pioglitazone/ja
Rivoglitazone/ja
†
Rosiglitazone/ja
Troglitazone/ja
‡
デュアルPPAR作動薬
Aleglitazar/ja
†
Muraglitazar/ja
§
Saroglitazar/ja
Tesaglitazar/ja
§
Amylin/ja
アナログと
DACRA
Cagrilintide/ja
§
Pramlintide/ja
セクレタゴーグ
K
+
ATP
スルホニル尿素
第一世代
:
Acetohexamide/ja
Carbutamide/ja
Chlorpropamide/ja
Glycyclamide/ja
Metahexamide/ja
Tolazamide/ja
Tolbutamide/ja
第二世代
:
グリベンクラミド(グリブリド)
Glibornuride/ja
Glicaramide/ja
Gliclazide/ja
#
グリメピリド
Glipizide/ja
Gliquidone/ja
Glisoxepide/ja
Glyclopyramide/ja
Meglitinide/ja
/"グリニド系"
Mitiglinide/ja
Nateglinide/ja
Repaglinide/ja
GLP-1受容体作動薬
Albiglutide/ja
‡
Danuglipron/ja
†
デュラグルチド
Exenatide/ja
Liraglutide/ja
Lixisenatide/ja
Orforglipron/ja
§
Semaglutide/ja
Taspoglutide/ja
†
GLP1ポリアゴニストペプチド
Mazdutide/ja
(GLP-1/
GCGR
)
Retatrutide/ja
§
(GLP-1/GIP/GCGR)
Tirzepatide/ja
(GLP-1/GIP)
DPP-4 阻害薬
/"グリプチン"
Alogliptin/ja
Anagliptin/ja
Evogliptin/ja
Garvagliptin/ja
Gemigliptin/ja
Gosogliptin/ja
Linagliptin/ja
Melogliptin/ja
Omarigliptin/ja
Saxagliptin/ja
シタグリプチン
Teneligliptin/ja
Trelagliptin/ja
Vildagliptin/ja
その他
Aldose reductase inhibitor/ja
Epalrestat/ja
Fidarestat/ja
§
Ranirestat/ja
†
Tolrestat/ja
‡
Zenarestat/ja
§
Alpha-glucosidase inhibitor/ja
Acarbose/ja
Miglitol/ja
Voglibose/ja
SGLT2 阻害薬
/"グリフロジン"
Canagliflozin/ja
Dapagliflozin/ja
Empagliflozin/ja
#
Ertugliflozin/ja
イプラグリフロジン
Luseogliflozin/ja
レモグリフロジン
§
セルグリフロジン
§
Sotagliflozin/ja
Tofogliflozin/ja
†
Velagliflozin/ja
その他
Benfluorex/ja
‡
Bromocriptine/ja
Imeglimin/ja
配合薬
Alogliptin/metformin/ja
Canagliflozin/metformin/ja
Cagrilintide/semaglutide/ja
§
Dapagliflozin/metformin/ja
Dapagliflozin/saxagliptin/ja
Dapagliflozin/saxagliptin/metformin/ja
Empagliflozin/linagliptin/ja
Empagliflozin/metformin/ja
Gemigliptin/rosuvastatin/ja
グリベンクラミド(グリブリド)/メトホルミン
Glimepiride/rosiglitazone/ja
Linagliptin/metformin/ja
Metformin/acarbose/ja
Metformin/ertugliflozin/ja
Metformin/evogliptin/ja
Metformin/gemigliptin/ja
Metformin/repaglinide/ja
Metformin/sulfonylureas/ja
Metformin/teneligliptin/ja
Phenformin/sulfonylureas/ja
Pioglitazone/alogliptin/ja
Pioglitazone/glimepiride/ja
Pioglitazone/metformin/ja
Pioglitazone/sitagliptin/ja
Rosiglitazone/metformin/ja
Saxagliptin/metformin/ja
Sitagliptin/dapagliflozin/ja
Sitagliptin/ertugliflozin/ja
Sitagliptin/metformin/ja
シタグリプチン/シンバスタチン
Vildagliptin/metformin/ja
#
WHO-EM
‡
Withdrawn
from market
Clinical trials
:
†
Phase III
§
Never to phase III
Portal
:
Medicine