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Discovery and development of gliflozins/36/en
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Drug design
Steps in design
Drug discovery
Hit to lead
Drug development
Preclinical
Clinical
Phases
Case studies of discovery
and development of drug classes
5α-Reductase inhibitors
ACE inhibitors
Angiotensin receptor blockers
Antiandrogens
Beta-blockers
Beta
2
agonists
Cephalosporins
c-Met inhibitors
Cyclooxygenase 2 inhibitors
Dipeptidyl peptidase-4 inhibitors
Direct thrombin inhibitors
Direct Xa inhibitors
Dual serotonin and norepinephrine reuptake inhibitors
Selective serotonin reuptake inhibitors
Gliflozins
HIV-protease inhibitors
Integrase inhibitors
Lipase inhibitors
Memantine and related drugs
mTOR inhibitors
Neuraminidase inhibitors
Non-nucleoside reverse-transcriptase inhibitors
NS5A inhibitors
Nucleoside and nucleotide reverse-transcriptase inhibitors
PDE5 inhibitors
Proton pump inhibitors
Statins
Thalidomide and its analogs
Triptans
TRPV1 antagonists
Tubulin inhibitors
Bcr-Abl tyrosine-kinase inhibitors
Cannabinoid receptor antagonists
CCR5 receptor antagonists
Neurokinin 1 receptor antagonists
5-HT
3
antagonists
Melatonin receptor agonists
Renin inhibitors