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Discovery and development of angiotensin receptor blockers/45/en
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t
e
Drug design
Steps in design
Drug discovery
Hit to lead
Drug development
Preclinical
Clinical
Phases
Case studies of discovery
and development of drug classes
5α-Reductase inhibitors
ACE inhibitors
Angiotensin receptor blockers
Antiandrogens
Beta-blockers
Beta
2
agonists
Cephalosporins
c-Met inhibitors
Cyclooxygenase 2 inhibitors
Dipeptidyl peptidase-4 inhibitors
Direct thrombin inhibitors
Direct Xa inhibitors
Dual serotonin and norepinephrine reuptake inhibitors
Selective serotonin reuptake inhibitors
Gliflozins
HIV-protease inhibitors
Integrase inhibitors
Lipase inhibitors
Memantine and related drugs
mTOR inhibitors
Neuraminidase inhibitors
Non-nucleoside reverse-transcriptase inhibitors
NS5A inhibitors
Nucleoside and nucleotide reverse-transcriptase inhibitors
PDE5 inhibitors
Proton pump inhibitors
Statins
Thalidomide and its analogs
Triptans
TRPV1 antagonists
Tubulin inhibitors
Bcr-Abl tyrosine-kinase inhibitors
Cannabinoid receptor antagonists
CCR5 receptor antagonists
Neurokinin 1 receptor antagonists
5-HT
3
antagonists
Melatonin receptor agonists
Renin inhibitors
v
t
e
Angiotensin receptor
modulators
ATR
Tooltip Angiotensin receptor
Agonists:
Angiotensin II
Angiotensin III
Angiotensin IV
L-163,491
Saralasin
Antagonists:
Abitesartan
Azilsartan
Candesartan
Elisartan
Embusartan
Eprosartan
EXP-3174
Fimasartan
Forasartan
Irbesartan
Losartan
Milfasartan
Olmesartan
Olodanrigan
PD123319
Pomisartan
Pratosartan
Ripisartan
Saprisartan
Sparsentan
Tasosartan
Telmisartan
Valsartan
Zolasartan
ACE
inhibitors:
Alacepril
Benazepril
Captopril
Cilazapril
Delapril
Enalapril
Enalaprilat
Fosinopril
Gemopatrilat
Imidapril
Lisinopril
Moexipril
Omapatrilat
Perindopril
Quinapril
Quinaprilat
Ramipril
Rentiapril
Rescinnamine
Spirapril
Spiraprilat
Temocapril
Trandolapril
Zofenopril
Zofenoprilat
Renin inhibitors:
Aliskiren
Ciprokiren
Ditekiren
Enalkiren
Imarikiren
Pepstatin
Remikiren
Terlakiren
Zankiren
Propeptides:
Angiotensinogen
Angiotensin I
Combinations:
Amlodipine/valsartan
Olmesartan/amlodipine
Olmesartan/amlodipine/hydrochlorothiazide
Valsartan/hydrochlorothiazide
Valsartan/hydrochlorothiazide/amlodipine