compound which inhibits or antagonizes the biosynthesis or actions of proteases (endopeptidases).
2 statements, 0 sitelinks - 10:26, 12 March 2024
[[Dipeptidyl peptidase-4 inhibitors]] (DPP-4 inhibitors) are [[enzyme inhibitor]]s that inhibit the [[enzyme]] [[dipeptidyl peptida
...[structure activity relationship]] (SAR) for subsequent investigation. The inhibitors fall into two main classes, those that interact covalently with DPP-4 and t
...
32 KB (4,417 words) - 10:31, 12 March 2024
[[Dipeptidyl peptidase-4 inhibitors]] (DPP-4 inhibitors) are [[enzyme inhibitor]]s that inhibit the [[enzyme]] [[dipeptidyl peptida
...[structure activity relationship]] (SAR) for subsequent investigation. The inhibitors fall into two main classes, those that interact covalently with DPP-4 and t
...
33 KB (4,561 words) - 10:30, 12 March 2024
...t increase activity. Many therapeutic [[drug]]s and [[poison]]s are enzyme inhibitors. An enzyme's activity decreases markedly outside its optimal [[temperature]
*EC 3, [[Hydrolase]]s: catalyze the [[hydrolysis]] of various bonds
...
52 KB (7,533 words) - 19:19, 21 February 2024
...t increase activity. Many therapeutic [[drug]]s and [[poison]]s are enzyme inhibitors. An enzyme's activity decreases markedly outside its optimal [[temperature]
*EC 3, [[Hydrolase]]s: catalyze the [[hydrolysis]] of various bonds
...
54 KB (7,773 words) - 19:18, 21 February 2024
...endocannabinoid [[2-arachidonoylglycerol]] (2-AG) while [[fatty acid amide hydrolase]] (FAAH) mediates the metabolism of [[anandamide]] into [[arachidonic acid]
...
23 KB (3,137 words) - 10:38, 28 February 2024
...endocannabinoid [[2-arachidonoylglycerol]] (2-AG) while [[fatty acid amide hydrolase]] (FAAH) mediates the metabolism of [[anandamide]] into [[arachidonic acid]
...
24 KB (3,233 words) - 10:37, 28 February 2024
*EC 3, [[Hydrolase/ja|ヒドロラーゼ]]:様々な結合の[[hydrolysis/ja|加水分解]]を触媒する
...a|スタチン]]や、[[HIV/ja|HIV]]のような[[retroviral/ja|レトロウイルス]]感染の治療に用いられる[[protease inhibitors/ja|プロテアーゼ阻害剤]]がある。薬物として使用される不可逆的阻害剤の一般的な例は[[aspirin/ja|アスピリン]]であり、これは[[infl
...
64 KB (2,204 words) - 15:33, 22 February 2024
...f some drugs as [[substrate (chemistry)|substrates]] or [[enzyme inhibitor|inhibitors]] of enzymes involved in xenobiotic metabolism are a common reason for haza
* [[Epoxide hydrolase]]
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29 KB (3,729 words) - 12:12, 15 November 2023
...[protease]]s that digest proteins into amino acids, as well as [[glycoside hydrolase]]s that digest polysaccharides into simple sugars known as [[monosaccharide
...and their [[enzyme kinetics|kinetics]] and responses to [[enzyme inhibitor|inhibitors]] investigated. A parallel approach is to identify the small molecules in a
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54 KB (7,765 words) - 19:27, 22 January 2024
...[protease]]s that digest proteins into amino acids, as well as [[glycoside hydrolase]]s that digest polysaccharides into simple sugars known as [[monosaccharide
...and their [[enzyme kinetics|kinetics]] and responses to [[enzyme inhibitor|inhibitors]] investigated. A parallel approach is to identify the small molecules in a
...
55 KB (7,943 words) - 19:27, 22 January 2024