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	<id>https://wiki.tiffa.net/w/index.php?action=history&amp;feed=atom&amp;title=Template%3AIonotropic_glutamate_receptor_modulators</id>
	<title>Template:Ionotropic glutamate receptor modulators - Revision history</title>
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	<updated>2026-04-18T15:08:37Z</updated>
	<subtitle>Revision history for this page on the wiki</subtitle>
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		<id>https://wiki.tiffa.net/w/index.php?title=Template:Ionotropic_glutamate_receptor_modulators&amp;diff=140821&amp;oldid=prev</id>
		<title>Fire: Created page with &quot;{{Navbox  | name = Ionotropic glutamate receptor modulators  | title = Ionotropic glutamate receptor modulators  | state = {{{state&lt;includeonly&gt;|collapsed&lt;/includeonly&gt;}}}  | bodyclass = hlist  | groupstyle = text-align:center;   | group1 = {{abbrlink|AMPAR|α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid receptor}}  | list1 = * &#039;&#039;&#039;Agonists:&#039;&#039;&#039; &#039;&#039;Main site agonists:&#039;&#039; 5-Fluorowillardiine * Acromelic acid A|Acromelic acid (acromelate)...&quot;</title>
		<link rel="alternate" type="text/html" href="https://wiki.tiffa.net/w/index.php?title=Template:Ionotropic_glutamate_receptor_modulators&amp;diff=140821&amp;oldid=prev"/>
		<updated>2024-04-18T10:24:02Z</updated>

		<summary type="html">&lt;p&gt;Created page with &amp;quot;{{Navbox  | name = Ionotropic glutamate receptor modulators  | title = &lt;a href=&quot;/w/index.php?title=Ionotropic_glutamate_receptor&amp;amp;action=edit&amp;amp;redlink=1&quot; class=&quot;new&quot; title=&quot;Ionotropic glutamate receptor (page does not exist)&quot;&gt;Ionotropic glutamate receptor&lt;/a&gt; &lt;a href=&quot;/w/index.php?title=Receptor_modulator&amp;amp;action=edit&amp;amp;redlink=1&quot; class=&quot;new&quot; title=&quot;Receptor modulator (page does not exist)&quot;&gt;modulators&lt;/a&gt;  | state = {{{state&amp;lt;includeonly&amp;gt;|collapsed&amp;lt;/includeonly&amp;gt;}}}  | bodyclass = hlist  | groupstyle = text-align:center;   | group1 = {{abbrlink|AMPAR|α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid receptor}}  | list1 = * &amp;#039;&amp;#039;&amp;#039;Agonists:&amp;#039;&amp;#039;&amp;#039; &amp;#039;&amp;#039;Main site agonists:&amp;#039;&amp;#039; &lt;a href=&quot;/w/index.php?title=5-Fluorowillardiine&amp;amp;action=edit&amp;amp;redlink=1&quot; class=&quot;new&quot; title=&quot;5-Fluorowillardiine (page does not exist)&quot;&gt;5-Fluorowillardiine&lt;/a&gt; * Acromelic acid A|Acromelic acid (acromelate)...&amp;quot;&lt;/p&gt;
&lt;p&gt;&lt;b&gt;New page&lt;/b&gt;&lt;/p&gt;&lt;div&gt;{{Navbox&lt;br /&gt;
 | name = Ionotropic glutamate receptor modulators&lt;br /&gt;
 | title = [[Ionotropic glutamate receptor]] [[receptor modulator|modulator]]s&lt;br /&gt;
 | state = {{{state&amp;lt;includeonly&amp;gt;|collapsed&amp;lt;/includeonly&amp;gt;}}}&lt;br /&gt;
 | bodyclass = hlist&lt;br /&gt;
 | groupstyle = text-align:center;&lt;br /&gt;
&lt;br /&gt;
 | group1 = {{abbrlink|AMPAR|α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid receptor}}&lt;br /&gt;
 | list1 =&lt;br /&gt;
* &amp;#039;&amp;#039;&amp;#039;Agonists:&amp;#039;&amp;#039;&amp;#039; &amp;#039;&amp;#039;Main site agonists:&amp;#039;&amp;#039; [[5-Fluorowillardiine]]&lt;br /&gt;
* [[Acromelic acid A|Acromelic acid (acromelate)]]&lt;br /&gt;
* [[AMPA]]&lt;br /&gt;
* [[β-N-Oxalylamino-L-Alanine|BOAA]]&lt;br /&gt;
* [[Domoic acid]]&lt;br /&gt;
* [[Glutamate]]&lt;br /&gt;
* [[Ibotenic acid]]&lt;br /&gt;
* [[Proline]]&lt;br /&gt;
* [[Quisqualic acid]]&lt;br /&gt;
* [[Willardiine]]; &amp;#039;&amp;#039;Positive allosteric modulators:&amp;#039;&amp;#039; [[Aniracetam]]&lt;br /&gt;
* [[Cyclothiazide]]&lt;br /&gt;
* [[CX-516]]&lt;br /&gt;
* [[CX-546]]&lt;br /&gt;
* [[CX614|CX-614]]&lt;br /&gt;
* [[Farampator|Farampator (CX-691, ORG-24448)]]&lt;br /&gt;
* [[CX717|CX-717]]&lt;br /&gt;
* [[CX-1739]]&lt;br /&gt;
* [[CX-1942]]&lt;br /&gt;
* [[Diazoxide]]&lt;br /&gt;
* [[Hydrochlorothiazide|Hydrochlorothiazide (HCTZ)]]&lt;br /&gt;
* [[IDRA-21]]&lt;br /&gt;
* [[LY-392098]]&lt;br /&gt;
* [[LY-395153]]&lt;br /&gt;
* [[LY-404187]]&lt;br /&gt;
* [[LY-451646]]&lt;br /&gt;
* [[LY-503430]]&lt;br /&gt;
* [[Mibampator|Mibampator (LY-451395)]]&lt;br /&gt;
* [[Nooglutyl]]&lt;br /&gt;
* [[ORG-26576]]&lt;br /&gt;
* [[Oxiracetam]]&lt;br /&gt;
* [[PEPA (drug)|PEPA]]&lt;br /&gt;
* [[Pesampator|Pesampator (BIIB-104, PF-04958242)]]&lt;br /&gt;
* [[Piracetam]]&lt;br /&gt;
* [[Pramiracetam]]&lt;br /&gt;
* [[S-18986]]&lt;br /&gt;
* [[Tulrampator|Tulrampator (S-47445, CX-1632)]]&lt;br /&gt;
&lt;br /&gt;
* &amp;#039;&amp;#039;&amp;#039;Antagonists:&amp;#039;&amp;#039;&amp;#039; [[ACEA-1011]]&lt;br /&gt;
* [[ATPO]]&lt;br /&gt;
* [[Becampanel]]&lt;br /&gt;
* [[Caroverine]]&lt;br /&gt;
* [[CNQX]]&lt;br /&gt;
* [[Dasolampanel]]&lt;br /&gt;
* [[DNQX]]&lt;br /&gt;
* [[Fanapanel|Fanapanel (MPQX)]]&lt;br /&gt;
* [[gamma-D-Glutamylaminomethylsulfonic acid|GAMS]]&lt;br /&gt;
* [[Kaitocephalin]]&lt;br /&gt;
* [[Kynurenic acid]]&lt;br /&gt;
* [[Kynurenine]]&amp;lt;!--As a prodrug of kynurenic acid--&amp;gt;&lt;br /&gt;
* [[Licostinel|Licostinel (ACEA-1021)]]&lt;br /&gt;
* [[NBQX]]&lt;br /&gt;
* [[PNQX]]&lt;br /&gt;
* [[Selurampanel]]&lt;br /&gt;
* [[Tezampanel]]&lt;br /&gt;
* [[Theanine]]&lt;br /&gt;
* [[Topiramate]]&lt;br /&gt;
* [[YM90K]]&lt;br /&gt;
* [[Zonampanel]]; &amp;#039;&amp;#039;Negative allosteric modulators:&amp;#039;&amp;#039; [[Barbiturates]] (e.g., [[pentobarbital]], [[sodium thiopental]])&lt;br /&gt;
* [[Cyclopropane]]&lt;br /&gt;
* [[Enflurane]]&lt;br /&gt;
* [[Alcohol (drug)|Ethanol (alcohol)]]&lt;br /&gt;
* [[Evans blue (dye)|Evans blue]]&lt;br /&gt;
* [[GYKI 52466|GYKI-52466]]&lt;br /&gt;
* [[GYKI-53655]]&lt;br /&gt;
* [[Halothane]]&lt;br /&gt;
* [[Irampanel]]&lt;br /&gt;
* [[Isoflurane]]&lt;br /&gt;
* [[Perampanel]]&lt;br /&gt;
* [[Pregnenolone sulfate]]&lt;br /&gt;
* [[Sevoflurane]]&lt;br /&gt;
* [[Talampanel]]; &amp;#039;&amp;#039;Unknown/unsorted antagonists:&amp;#039;&amp;#039; [[Minocycline]]&lt;br /&gt;
&lt;br /&gt;
 | group2 = {{abbrlink|KAR|Kainate receptor}}&lt;br /&gt;
 | list2 =&lt;br /&gt;
* &amp;#039;&amp;#039;&amp;#039;Agonists:&amp;#039;&amp;#039;&amp;#039; &amp;#039;&amp;#039;Main site agonists:&amp;#039;&amp;#039; [[5-Bromowillardiine]]&lt;br /&gt;
* [[5-Iodowillardiine]]&lt;br /&gt;
* [[Acromelic acid|Acromelic acid (acromelate)]]&lt;br /&gt;
* [[AMPA]]&lt;br /&gt;
* [[ATPA]]&lt;br /&gt;
* [[Domoic acid]]&lt;br /&gt;
* [[Glutamate]]&lt;br /&gt;
* [[Ibotenic acid]]&lt;br /&gt;
* [[Kainic acid]]&lt;br /&gt;
* [[LY-339434]]&lt;br /&gt;
* [[Proline]]&lt;br /&gt;
* [[Quisqualic acid]]&lt;br /&gt;
* [[SYM-2081]]; &amp;#039;&amp;#039;Positive allosteric modulators:&amp;#039;&amp;#039; [[Cyclothiazide]]&lt;br /&gt;
* [[Diazoxide]]&lt;br /&gt;
* [[Enflurane]]&lt;br /&gt;
* [[Halothane]]&lt;br /&gt;
* [[Isoflurane]]&lt;br /&gt;
&lt;br /&gt;
* &amp;#039;&amp;#039;&amp;#039;Antagonists:&amp;#039;&amp;#039;&amp;#039; [[ACEA-1011]]&lt;br /&gt;
* [[CNQX]]&lt;br /&gt;
* [[Dasolampanel]]&lt;br /&gt;
* [[DNQX]]&lt;br /&gt;
* [[gamma-D-Glutamylaminomethylsulfonic acid|GAMS]]&lt;br /&gt;
* [[Kaitocephalin]]&lt;br /&gt;
* [[Kynurenic acid]]&lt;br /&gt;
* [[Licostinel|Licostinel (ACEA-1021)]]&lt;br /&gt;
* [[LY-382884]]&lt;br /&gt;
* [[NBQX]]&lt;br /&gt;
* [[NS102]]&lt;br /&gt;
* [[Selurampanel]]&lt;br /&gt;
* [[Tezampanel]]&lt;br /&gt;
* [[Theanine]]&lt;br /&gt;
* [[Topiramate]]&lt;br /&gt;
* [[UBP-302]]; &amp;#039;&amp;#039;Negative allosteric modulators:&amp;#039;&amp;#039; [[Barbiturates]] (e.g., [[pentobarbital]], [[sodium thiopental]])&lt;br /&gt;
* [[Enflurane]]&lt;br /&gt;
* [[Alcohol (drug)|Ethanol (alcohol)]]&lt;br /&gt;
* [[Evans blue (dye)|Evans blue]]&lt;br /&gt;
* [[NS-3763]]&lt;br /&gt;
* [[Pregnenolone sulfate]]&lt;br /&gt;
&lt;br /&gt;
 | group3 = {{abbrlink|NMDAR|N-Methyl-D-aspartate receptor}}&lt;br /&gt;
 | list3 =&lt;br /&gt;
* &amp;#039;&amp;#039;&amp;#039;Agonists:&amp;#039;&amp;#039;&amp;#039; &amp;#039;&amp;#039;Main site agonists:&amp;#039;&amp;#039; [[2-Amino-2-(3-hydroxy-5-methylisoxazol-4-yl)acetic acid|AMAA]]&lt;br /&gt;
* [[Aspartate]]&lt;br /&gt;
* [[Glutamate]]&lt;br /&gt;
* [[Homocysteic acid|Homocysteic acid (&amp;lt;small&amp;gt;L&amp;lt;/small&amp;gt;-HCA)]]&lt;br /&gt;
* [[Homoquinolinic acid]]&lt;br /&gt;
* [[Ibotenic acid]]&lt;br /&gt;
* [[N-Methyl-D-aspartic acid|NMDA]]&lt;br /&gt;
* [[Proline]]&lt;br /&gt;
* [[Quinolinic acid]]&lt;br /&gt;
* [[Tetrazolylglycine]]&lt;br /&gt;
* [[Theanine]]; &amp;#039;&amp;#039;Glycine site agonists:&amp;#039;&amp;#039; [[β-Fluoro-D-alanine|β-Fluoro-&amp;lt;small&amp;gt;D&amp;lt;/small&amp;gt;-alanine]]&lt;br /&gt;
* [[ACBD (drug)|ACBD]]&lt;br /&gt;
* [[1-Aminocyclopropanecarboxylic acid|ACC (ACPC)]]&lt;br /&gt;
* [[ACPD]]&lt;br /&gt;
* [[AK-51 (drug)|AK-51]]&lt;br /&gt;
* [[Apimostinel|Apimostinel (NRX-1074)]]&lt;br /&gt;
* [[B6B21]]&lt;br /&gt;
* [[Carboxycyclopropylglycine|CCG]]&lt;br /&gt;
* [[Alanine|&amp;lt;small&amp;gt;D&amp;lt;/small&amp;gt;-Alanine]]&lt;br /&gt;
* [[Cycloserine|&amp;lt;small&amp;gt;D&amp;lt;/small&amp;gt;-Cycloserine]]&lt;br /&gt;
* [[Serine|&amp;lt;small&amp;gt;D&amp;lt;/small&amp;gt;-Serine]]&lt;br /&gt;
* [[N-(3,3-Diphenylpropyl)glycinamide|DHPG]]&lt;br /&gt;
* [[Dimethylglycine]]&lt;br /&gt;
* [[Glycine]]&lt;br /&gt;
* [[HA-966]]&lt;br /&gt;
* [[L-687414]]&lt;br /&gt;
* [[Alanine|&amp;lt;small&amp;gt;L&amp;lt;/small&amp;gt;-Alanine]]&lt;br /&gt;
* [[Serine|&amp;lt;small&amp;gt;L&amp;lt;/small&amp;gt;-Serine]]&lt;br /&gt;
* [[Milacemide]]&lt;br /&gt;
* [[Neboglamine|Neboglamine (nebostinel)]]&lt;br /&gt;
* [[Rapastinel|Rapastinel (GLYX-13)]]&lt;br /&gt;
* [[Sarcosine]]; &amp;#039;&amp;#039;Polyamine site agonists:&amp;#039;&amp;#039; [[Neomycin]]&lt;br /&gt;
* [[Spermidine]]&lt;br /&gt;
* [[Spermine]]; &amp;#039;&amp;#039;Other positive allosteric modulators:&amp;#039;&amp;#039; [[24S-Hydroxycholesterol|24&amp;#039;&amp;#039;S&amp;#039;&amp;#039;-Hydroxycholesterol]]&lt;br /&gt;
* {{abbrlink|DHEA|Dehydroepiandrosterone}} ([[prasterone]])&lt;br /&gt;
* [[Dehydroepiandrosterone sulfate|{{abbr|DHEA|Dehydroepiandrosterone}} sulfate]] ([[prasterone sulfate]])&lt;br /&gt;
* [[Epipregnanolone sulfate]]&lt;br /&gt;
* [[Plazinemdor]]&lt;br /&gt;
* [[Pregnenolone sulfate]]&lt;br /&gt;
* [[SAGE-201]]&lt;br /&gt;
* [[SAGE-301]]&lt;br /&gt;
* [[SAGE-718]]&lt;br /&gt;
&lt;br /&gt;
* &amp;#039;&amp;#039;&amp;#039;Antagonists:&amp;#039;&amp;#039;&amp;#039; &amp;#039;&amp;#039;Competitive antagonists:&amp;#039;&amp;#039; [[AP5|AP5 (APV)]]&lt;br /&gt;
* [[AP-7 (drug)|AP7]]&lt;br /&gt;
* [[CGP-37849]]&lt;br /&gt;
* [[CGP-39551]]&lt;br /&gt;
* [[CGP-39653]]&lt;br /&gt;
* [[CGP-40116]]&lt;br /&gt;
* [[CGS-19755]]&lt;br /&gt;
* [[3-(2-carboxypiperazin-4-yl)propyl-1-phosphonic acid|CPP]]&lt;br /&gt;
* [[Kaitocephalin]]&lt;br /&gt;
* [[LY-233053]]&lt;br /&gt;
* [[LY-235959]]&lt;br /&gt;
* [[LY-274614]]&lt;br /&gt;
* [[MDL-100453]]&lt;br /&gt;
* [[Midafotel|Midafotel (d-CPPene)]]&lt;br /&gt;
* [[NPC-12626]]&lt;br /&gt;
* [[NPC-17742]]&lt;br /&gt;
* [[PBPD]]&lt;br /&gt;
* [[PEAQX]]&lt;br /&gt;
* [[Perzinfotel]]&lt;br /&gt;
* [[cis-1-(phenanthrene-2-carbonyl)piperazine-2,3-dicarboxylic acid|PPDA]]&lt;br /&gt;
* [[SDZ-220581]]&lt;br /&gt;
* [[Selfotel]]; &amp;#039;&amp;#039;Glycine site antagonists:&amp;#039;&amp;#039; [[4-Chlorokynurenine|4-Cl-KYN (AV-101)]]&lt;br /&gt;
* [[5,7-Dichlorokynurenic acid|5,7-DCKA]]&lt;br /&gt;
* [[7-Chlorokynurenic acid|7-CKA]]&lt;br /&gt;
* [[1-Aminocyclopropane-1-carboxylic acid|ACC]]&lt;br /&gt;
* [[ACEA-1011]]&lt;br /&gt;
* [[ACEA-1328]]&lt;br /&gt;
* [[Apimostinel|Apimostinel (NRX-1074)]]&lt;br /&gt;
* [[AV-101]]&lt;br /&gt;
* [[Carisoprodol]]&lt;br /&gt;
* [[CGP-39653]]&lt;br /&gt;
* [[CNQX]]&lt;br /&gt;
* [[Cycloserine|&amp;lt;small&amp;gt;D&amp;lt;/small&amp;gt;-Cycloserine]]&lt;br /&gt;
* [[DNQX]]&lt;br /&gt;
* [[Felbamate]]&lt;br /&gt;
* [[Gavestinel]]&lt;br /&gt;
* [[GV-196771]]&lt;br /&gt;
* [[Harkoseride]]&lt;br /&gt;
* [[Kynurenic acid]]&lt;br /&gt;
* [[Kynurenine]]&amp;lt;!--As a prodrug of kynurenic acid--&amp;gt;&lt;br /&gt;
* [[L-689560]]&lt;br /&gt;
* [[L-701324]]&lt;br /&gt;
* [[Licostinel|Licostinel (ACEA-1021)]]&lt;br /&gt;
* [[LU-73068]]&lt;br /&gt;
* [[MDL-105519]]&lt;br /&gt;
* [[Meprobamate]]&lt;br /&gt;
* [[MRZ 2/576]]&lt;br /&gt;
* [[PNQX]]&lt;br /&gt;
* [[Rapastinel|Rapastinel (GLYX-13)]]&lt;br /&gt;
* [[ZD-9379]]; &amp;#039;&amp;#039;Polyamine site antagonists:&amp;#039;&amp;#039; [[Arcaine]]&lt;br /&gt;
* [[Co 101676]]&lt;br /&gt;
* [[1,3-Diaminopropane|Diaminopropane]]&lt;br /&gt;
* [[Diethylenetriamine]]&lt;br /&gt;
* [[Huperzine A]]&lt;br /&gt;
* [[Putrescine]]; &amp;#039;&amp;#039;Uncompetitive pore blockers (mostly dizocilpine site):&amp;#039;&amp;#039; [[2-MDP]]&lt;br /&gt;
* [[3-HO-PCP]]&lt;br /&gt;
* [[3-MeO-PCE]]&lt;br /&gt;
* [[3-MeO-PCMo]]&lt;br /&gt;
* [[3-MeO-PCP]]&lt;br /&gt;
* [[4-MeO-PCP]]&lt;br /&gt;
* [[8a-Phenyldecahydroquinoline|8A-PDHQ]]&lt;br /&gt;
* [[18-Methoxycoronaridine|18-MC]]&lt;br /&gt;
* [[Alpha-Endopsychosin|α-Endopsychosin]]&lt;br /&gt;
* [[Alaproclate]]&lt;br /&gt;
* [[Alazocine|Alazocine (SKF-10047)]]&lt;br /&gt;
* [[Amantadine]]&lt;br /&gt;
* [[Aptiganel]]&lt;br /&gt;
* [[Argiotoxin-636]]&lt;br /&gt;
* [[Arketamine]]&lt;br /&gt;
* [[ARL-12495]]&lt;br /&gt;
* [[ARL-15896-AR]]&lt;br /&gt;
* [[ARL-16247]]&lt;br /&gt;
* [[Budipine]]&lt;br /&gt;
* [[Coronaridine]]&lt;br /&gt;
* [[Delucemine|Delucemine (NPS-1506)]]&lt;br /&gt;
* [[Dexoxadrol]]&lt;br /&gt;
* [[Dextrallorphan]]&lt;br /&gt;
* [[Dextromethadone]]&lt;br /&gt;
* [[Dextromethorphan]]&lt;br /&gt;
* [[Dextrorphan]]&lt;br /&gt;
* [[Dieticyclidine]]&lt;br /&gt;
* [[Diphenidine]]&lt;br /&gt;
* [[Dizocilpine]]&lt;br /&gt;
* [[Ephenidine]]&lt;br /&gt;
* [[Esketamine]]&lt;br /&gt;
* [[Etoxadrol]]&lt;br /&gt;
* [[Eticyclidine]]&lt;br /&gt;
* [[Fluorolintane]]&lt;br /&gt;
* [[Gacyclidine]]&lt;br /&gt;
* [[Ibogaine]]&lt;br /&gt;
* [[Ibogamine]]&lt;br /&gt;
* [[Indantadol]]&lt;br /&gt;
* [[Ketamine]]&lt;br /&gt;
* [[Ketobemidone]]&lt;br /&gt;
* [[Lanicemine]]&lt;br /&gt;
* [[Levomethadone]]&lt;br /&gt;
* [[Levomethorphan]]&lt;br /&gt;
* [[Levomilnacipran]]&lt;br /&gt;
* [[Levorphanol]]&lt;br /&gt;
* [[Loperamide]]&lt;br /&gt;
* [[Memantine]]&lt;br /&gt;
* [[Methadone]]&lt;br /&gt;
* [[Methorphan]]&lt;br /&gt;
* [[Methoxetamine]]&lt;br /&gt;
* [[Methoxphenidine]]&lt;br /&gt;
* [[Milnacipran]]&lt;br /&gt;
* [[Morphanol]]&lt;br /&gt;
* [[NEFA (drug)|NEFA]]&lt;br /&gt;
* [[Neramexane]]&lt;br /&gt;
* [[Nitromemantine]]&lt;br /&gt;
* [[Noribogaine]]&lt;br /&gt;
* [[Norketamine]]&lt;br /&gt;
* [[Orphenadrine]]&lt;br /&gt;
* [[PCPr]]&lt;br /&gt;
* [[PD-137889]]&lt;br /&gt;
* [[Pethidine|Pethidine (meperidine)]]&lt;br /&gt;
* [[Phencyclamine]]&lt;br /&gt;
* [[Phencyclidine]]&lt;br /&gt;
* [[Propoxyphene]]&lt;br /&gt;
* [[Remacemide]]&lt;br /&gt;
* [[Rhynchophylline]]&lt;br /&gt;
* [[Rimantadine]]&lt;br /&gt;
* [[Rolicyclidine]]&lt;br /&gt;
* [[Sabeluzole]]&lt;br /&gt;
* [[Tabernanthine]]&lt;br /&gt;
* [[Tenocyclidine]]&lt;br /&gt;
* [[Tiletamine]]&lt;br /&gt;
* [[Tramadol]]; &amp;#039;&amp;#039;Ifenprodil (NR2B) site antagonists:&amp;#039;&amp;#039;&lt;br /&gt;
* [[Besonprodil]]&lt;br /&gt;
* [[Buphenine|Buphenine (nylidrin)]]&lt;br /&gt;
* [[CO-101244|CO-101244 (PD-174494)]]&lt;br /&gt;
* [[Eliprodil]]&lt;br /&gt;
* [[Haloperidol]]&lt;br /&gt;
* [[Isoxsuprine]]&lt;br /&gt;
* [[Radiprodil|Radiprodil (RGH-896)]]&lt;br /&gt;
* [[Rislenemdaz|Rislenemdaz (CERC-301, MK-0657)]]&lt;br /&gt;
* [[Ro 8-4304]]&lt;br /&gt;
* [[Ro 25-6981]]&lt;br /&gt;
* [[Safaprodil]]&lt;br /&gt;
* [[Traxoprodil|Traxoprodil (CP-101606)]]; &amp;#039;&amp;#039;NR2A-selective antagonists:&amp;#039;&amp;#039; [[MPX-004]]&lt;br /&gt;
* [[MPX-007]]&lt;br /&gt;
* [[TCN-201]]&lt;br /&gt;
* [[TCN-213]]; &amp;#039;&amp;#039;Cations:&amp;#039;&amp;#039; [[Hydrogen]]&lt;br /&gt;
* [[Magnesium]]&lt;br /&gt;
* [[Zinc]]; &amp;#039;&amp;#039;Alcohols/volatile anesthetics/related:&amp;#039;&amp;#039; [[Benzene]]&lt;br /&gt;
* [[Butane]]&lt;br /&gt;
* [[Chloroform]]&lt;br /&gt;
* [[Cyclopropane]]&lt;br /&gt;
* [[Desflurane]]&lt;br /&gt;
* [[Diethyl ether]]&lt;br /&gt;
* [[Enflurane]]&lt;br /&gt;
* [[Alcohol (drug)|Ethanol (alcohol)]]&lt;br /&gt;
* [[Halothane]]&lt;br /&gt;
* [[Hexanol]]&lt;br /&gt;
* [[Isoflurane]]&lt;br /&gt;
* [[Methoxyflurane]]&lt;br /&gt;
* [[Nitrous oxide]]&lt;br /&gt;
* [[Octanol]]&lt;br /&gt;
* [[Sevoflurane]]&lt;br /&gt;
* [[Toluene]]&lt;br /&gt;
* [[1,1,1-Trichloroethane|Trichloroethane]]&lt;br /&gt;
* [[2,2,2-Trichloroethanol|Trichloroethanol]]&lt;br /&gt;
* [[Trichloroethylene]]&lt;br /&gt;
* [[Ethyl carbamate|Urethane]]&lt;br /&gt;
* [[Xenon]]&lt;br /&gt;
* [[Xylene]]; &amp;#039;&amp;#039;Unknown/unsorted antagonists:&amp;#039;&amp;#039; [[ARR-15896]]&lt;br /&gt;
* [[Bumetanide]]&lt;br /&gt;
* [[Caroverine]]&lt;br /&gt;
* [[Conantokin]]&lt;br /&gt;
* [[D-α-Aminoadipate|&amp;lt;small&amp;gt;D&amp;lt;/small&amp;gt;-αAA]]&lt;br /&gt;
* [[Dexanabinol]]&lt;br /&gt;
* [[Flufenamic acid]]&lt;br /&gt;
* [[Flupirtine]]&lt;br /&gt;
* [[FPL-12495]]&lt;br /&gt;
* [[FR-115427]]&lt;br /&gt;
* [[Furosemide]]&lt;br /&gt;
* [[Hodgkinsine]]&lt;br /&gt;
* [[Ipenoxazone|Ipenoxazone (MLV-6976)]]&lt;br /&gt;
* [[MDL-27266]]&lt;br /&gt;
* [[Metaphit]]&amp;lt;!--Irreversible--&amp;gt;&lt;br /&gt;
* [[Minocycline]]&lt;br /&gt;
* [[2-Methyl-6-(phenylethynyl)pyridine|MPEP]]&lt;br /&gt;
* [[Niflumic acid]]&lt;br /&gt;
* [[Pentamidine]]&lt;br /&gt;
* [[Pentamidine isethionate]]&lt;br /&gt;
* [[Piretanide]]&lt;br /&gt;
* [[Psychotridine]]&lt;br /&gt;
* [[Transcrocetin]] ([[saffron]])&lt;br /&gt;
&lt;br /&gt;
* &amp;#039;&amp;#039;&amp;#039;Unsorted:&amp;#039;&amp;#039;&amp;#039; &amp;#039;&amp;#039;Allosteric modulators:&amp;#039;&amp;#039; [[AGN-241751]]&lt;br /&gt;
&lt;br /&gt;
|below =&lt;br /&gt;
* &amp;#039;&amp;#039;&amp;#039;&amp;#039;&amp;#039;See also:&amp;#039;&amp;#039;&amp;#039; [[Template:Receptor modulators|Receptor/signaling modulators]]&amp;#039;&amp;#039;&lt;br /&gt;
* &amp;#039;&amp;#039;[[Template:Metabotropic glutamate receptor modulators|Metabotropic glutamate receptor modulators]]&amp;#039;&amp;#039;&lt;br /&gt;
* &amp;#039;&amp;#039;[[Template:Glutamate metabolism and transport modulators|Glutamate metabolism/transport modulators]]&amp;#039;&amp;#039;&lt;br /&gt;
}}&lt;br /&gt;
&amp;lt;noinclude&amp;gt;&lt;br /&gt;
{{Collapsible option}}&lt;br /&gt;
[[Category:Drug templates by receptor, channel, or pump]]&lt;br /&gt;
&amp;lt;/noinclude&amp;gt;&lt;/div&gt;</summary>
		<author><name>Fire</name></author>
	</entry>
</feed>